Llwytho...

Binding of RyR2 “Unzipping” Peptide in Cardiomyocytes Activates RyR2 and Reciprocally Inhibits Calmodulin Binding

RATIONALE: One hypothesis for elevated Ca(2+) leak through cardiac ryanodine receptors (RyR2) in heart failure (HF) is interdomain “unzipping” that can enhance aberrant channel activation. A peptide (DPc10) corresponding to RyR2 central domain 2460-2495 recapitulates this arrhythmogenic RyR2 leakine...

Disgrifiad llawn

Wedi'i Gadw mewn:
Manylion Llyfryddiaeth
Prif Awduron: Oda, Tetsuro, Yang, Yi, Nitu, Florentin R., Svensson, Bengt, Lu, Xiyuan, Fruen, Bradley R., Cornea, Razvan L., Bers, Donald M.
Fformat: Artigo
Iaith:Inglês
Cyhoeddwyd: 2012
Pynciau:
Mynediad Ar-lein:https://ncbi.nlm.nih.gov/pmc/articles/PMC3573756/
https://ncbi.nlm.nih.gov/pubmed/23233753
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1161/CIRCRESAHA.111.300290
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