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4′-Methyl-4,5′-bithiazole-based correctors of defective ΔF508-CFTR cellular processing

The synthesis and ΔF508-CFTR corrector activity of a 148-member methylbithiazole-based library is reported. Synthetic routes were devised and optimized to generate methylbithiazole analogs in four steps. Corrector potency and efficacy was assayed using epithelial cells expressing human ΔF508-CFTR. T...

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Autores principales: Yoo, Choong Leol, Yu, Gui Jun, Yang, Baoxue, Robins, Lori I., Verkman, A.S., Kurth, Mark J.
Formato: Artigo
Lenguaje:Inglês
Publicado: 2008
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC3166558/
https://ncbi.nlm.nih.gov/pubmed/18394886
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmcl.2008.03.037
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