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Inhibition of β-Secretase in Vivo via Antibody Binding to Unique Loops (D and F) of BACE1

β-Secretase (BACE1) is an attractive drug target for Alzheimer disease. However, the design of clinical useful inhibitors targeting its active site has been extremely challenging. To identify alternative drug targeting sites we have generated a panel of BACE1 monoclonal antibodies (mAbs) that interf...

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Gorde:
Xehetasun bibliografikoak
Egile Nagusiak: Zhou, Lujia, Chávez-Gutiérrez, Lucia, Bockstael, Katrijn, Sannerud, Ragna, Annaert, Wim, May, Patrick C., Karran, Eric, De Strooper, Bart
Formatua: Artigo
Hizkuntza:Inglês
Argitaratua: American Society for Biochemistry and Molecular Biology 2011
Gaiak:
Sarrera elektronikoa:https://ncbi.nlm.nih.gov/pmc/articles/PMC3048749/
https://ncbi.nlm.nih.gov/pubmed/21209097
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1074/jbc.M110.194860
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