Novel synthetic route to the C-nucleoside, 2-deoxy benzamide riboside

по Midtkandal, Rebecca R., Redpath, Philip, Trammell, Samuel A.J., Macdonald, Simon J.F., Brenner, Charles, Migaud, Marie E.
Опубликовано 2012

Relative Binding Affinities of Integrin Antagonists by Equilibrium Dialysis and Liquid Chromatography–Mass Spectrometry

по Tipping, William J., Tshuma, Nkazimulo, Adams, James, Haywood, Harvey T., Rowedder, James E., Fray, M. Jonathan, McInally, Thomas, Macdonald, Simon J. F., Oldham, Neil J.
Опубликовано в: ACS Med Chem Lett (2014)

An Invitation to Open Innovation in Malaria Drug Discovery: 47 Quality Starting Points from the TCAMS

по Calderón, Félix, Barros, David, Bueno, José María, Coterón, José Miguel, Fernández, Esther, Gamo, Francisco Javier, Lavandera, José Luís, León, María Luisa, Macdonald, Simon J. F., Mallo, Araceli, Manzano, Pilar, Porras, Esther, Fiandor, José María, Castro, Julia
Опубликовано 2011

Cyclopropyl Carboxamides: A New Oral Antimalarial Series Derived from the Tres Cantos Anti-Malarial Set (TCAMS)

по Rueda, Lourdes, Castellote, Isabel, Castro-Pichel, Julia, Chaparro, Maria J., de la Rosa, Juan Carlos, Garcia-Perez, Adolfo, Gordo, Mariola, Jimenez-Diaz, Maria Belen, Kessler, Albane, Macdonald, Simon J.F., Martinez, Maria Santos, Sanz, Laura M., Gamo, Francisco Javier, Fernandez, Esther
Опубликовано 2011

Design and x-ray crystal structures of high-potency nonsteroidal glucocorticoid agonists exploiting a novel binding site on the receptor

по Biggadike, Keith, Bledsoe, Randy K., Coe, Diane M., Cooper, Tony W. J., House, David, Iannone, Marie A., Macdonald, Simon J. F., Madauss, Kevin P., McLay, Iain M., Shipley, Tracy J., Taylor, Simon J., Tran, Thuy B., Uings, Iain J., Weller, Victoria, Williams, Shawn P.
Опубликовано 2009

Structure Activity Relationships of α(v) Integrin Antagonists for Pulmonary Fibrosis by Variation in Aryl Substituents

по Adams, James, Anderson, Edward C., Blackham, Emma E., Chiu, Yin Wa Ryan, Clarke, Thomas, Eccles, Natasha, Gill, Luke A., Haye, Joshua J., Haywood, Harvey T., Hoenig, Christian R., Kausas, Marius, Le, Joelle, Russell, Hannah L., Smedley, Christopher, Tipping, William J., Tongue, Tom, Wood, Charlotte C., Yeung, Jason, Rowedder, James E., Fray, M. Jonathan, McInally, Thomas, Macdonald, Simon J. F.
Опубликовано в: ACS Med Chem Lett (2014)

Potent and Long-Acting Dimeric Inhibitors of Influenza Virus Neuraminidase Are Effective at a Once-Weekly Dosing Regimen

по Macdonald, Simon J. F., Watson, Keith G., Cameron, Rachel, Chalmers, David K., Demaine, Derek A., Fenton, Rob J., Gower, David, Hamblin, J. Nicole, Hamilton, Stephanie, Hart, Graham J., Inglis, Graham G. A., Jin, Betty, Jones, Haydn T., McConnell, Darryl B., Mason, Andy M., Nguyen, Van, Owens, Ian J., Parry, Nigel, Reece, Phillip A., Shanahan, Stephen E., Smith, Donna, Wu, Wen-Yang, Tucker, Simon P.
Опубликовано 2004

Translational pharmacology of an inhaled small molecule αvβ6 integrin inhibitor for idiopathic pulmonary fibrosis

по John, Alison E., Graves, Rebecca H., Pun, K. Tao, Vitulli, Giovanni, Forty, Ellen J., Mercer, Paul F., Morrell, Josie L., Barrett, John W., Rogers, Rebecca F., Hafeji, Maryam, Bibby, Lloyd I., Gower, Elaine, Morrison, Valerie S., Man, Yim, Roper, James A., Luckett, Jeni C., Borthwick, Lee A., Barksby, Ben S., Burgoyne, Rachel A., Barnes, Rory, Le, Joelle, Flint, David J., Pyne, Susan, Habgood, Anthony, Organ, Louise A., Joseph, Chitra, Edwards-Pritchard, Rochelle C., Maher, Toby M., Fisher, Andrew J., Gudmann, Natasja Stæhr, Leeming, Diana J., Chambers, Rachel C., Lukey, Pauline T., Marshall, Richard P., Macdonald, Simon J. F., Jenkins, R. Gisli, Slack, Robert J.
Опубликовано в: Nat Commun (2020)