Small Molecule Modulation of Nuclear Receptor Conformational Dynamics: Implications for Function and Drug Discovery

od Kojetin, Douglas J., Burris, Thomas P.
Izdano 2013

REV-ERB and ROR nuclear receptors as drug targets

od Kojetin, Douglas J., Burris, Thomas P.
izdano v Nat Rev Drug Discov (2014)

Anti-Proliferative Actions of a Synthetic REV-ERBα/β Agonist in Breast Cancer Cells

od Wang, Yongjun, Kojetin, Douglas, Burris, Thomas P.
izdano v Biochem Pharmacol (2015)

The REV-ERBs and RORs: molecular links between circadian rhythms and lipid homeostasis

od Solt, Laura A, Kojetin, Douglas J, Burris, Thomas P
Izdano 2011

Characterization of the Core Mammalian Clock Component, NPAS2, as a REV-ERBα/RORα Target Gene

od Crumbley, Christine, Wang, Yongjun, Kojetin, Douglas J., Burris, Thomas P.
Izdano 2010

Identification of SR8278, a Synthetic Antagonist of the Nuclear Heme Receptor REV-ERB

od Kojetin, Douglas, Wang, Yongjun, Kameneck, Theodore M., Burris, Thomas P.
Izdano 2010

Activity-based profiling reveals a regulatory link between oxidative stress and protein arginine phosphorylation

od Fuhrmann, Jakob, Subramanian, Venkataraman, Kojetin, Douglas J., Thompson, Paul R.
izdano v Cell Chem Biol (2016)

(1)H, (13)C and (15)N chemical shift assignments for the human Pitx2 homeodomain and a R24H homeodomain mutant

od Doerdelmann, Thomas, Kojetin, Douglas J., Baird-Titus, Jamie M., Rance, Mark
Izdano 2010

(1)H, (13)C and (15)N chemical shift assignments for the human Pitx2 homeodomain in complex with a 22-base hairpin DNA

od Doerdelmann, Thomas, Kojetin, Douglas J., Baird-Titus, Jamie M., Rance, Mark
Izdano 2011

Regulation of p53 Stability and Apoptosis by a ROR Agonist

od Wang, Yongjun, Solt, Laura A., Kojetin, Douglas J., Burris, Thomas P.
Izdano 2012

Alternative Splicing of a β(4) Subunit Proline-Rich Motif Regulates Voltage-Dependent Gating and Toxin Block of Ca(v)2.1 Ca(2+) Channels

od Helton, Thomas D., Kojetin, Douglas J., Cavanagh, John, Horne, William A.
izdano v J Neurosci (2002)

Deconvolution of Complex 1D NMR Spectra Using Objective Model Selection

od Hughes, Travis S., Wilson, Henry D., de Vera, Ian Mitchelle S., Kojetin, Douglas J.
izdano v PLoS One (2015)

Quantitative structural assessment of graded receptor agonism

od Shang, Jinsai, Brust, Richard, Griffin, Patrick R., Kamenecka, Theodore M., Kojetin, Douglas J.
izdano v Proc Natl Acad Sci U S A (2019)

Modification of the Orthosteric PPARγ Covalent Antagonist Scaffold Yields an Improved Dual-Site Allosteric Inhibitor

od Brust, Richard, Lin, Hua, Fuhrmann, Jakob, Asteian, Alice, Kamenecka, Theodore M., Kojetin, Douglas J.
izdano v ACS Chem Biol (2017)

Structural and Biophysical Insights into the Ligand-Free Pitx2 Homeodomain and a Ring Dermoid of the Cornea Inducing Homeodomain Mutant

od Doerdelmann, Thomas, Kojetin, Douglas J., Baird-Titus, Jamie M., Solt, Laura A., Burris, Thomas P., Rance, Mark
Izdano 2012

Assessment of NR4A Ligands that Directly Bind and Modulate the Orphan Nuclear Receptor Nurr1

od Munoz-Tello, Paola, Lin, Hua, Khan, Pasha, de Vera, Ian Mitchelle S., Kamenecka, Theodore M., Kojetin, Douglas J.
izdano v J Med Chem (2020)

Structural and motional contributions of the Bacillus subtilis ClpC N-domain in adaptor protein interactions

od Kojetin, Douglas J., McLaughlin, Patrick D., Thompson, Richele J., Dubnau, David, Prepiak, Peter, Rance, Mark, Cavanagh, John
Izdano 2009

Observing selected domains in multi-domain proteins via sortase-mediated ligation and NMR spectroscopy

od Refaei, Mary Anne, Combs, Al, Kojetin, Douglas J., Cavanagh, John, Caperelli, Carol, Rance, Mark, Sapitro, Jennifer, Tsang, Pearl
Izdano 2010

Structure of REV-ERBβ Ligand-binding Domain Bound to a Porphyrin Antagonist

od Matta-Camacho, Edna, Banerjee, Subhashis, Hughes, Travis S., Solt, Laura A., Wang, Yongjun, Burris, Thomas P., Kojetin, Douglas J.
Izdano 2014

Insights into the nature of DNA binding of AbrB-like transcription factors

od Sullivan, Daniel M., Bobay, Benjamin G., Kojetin, Douglas J., Thompson, Richele J., Rance, Mark, Strauch, Mark A., Cavanagh, John
Izdano 2008