Small Molecule Modulation of Nuclear Receptor Conformational Dynamics: Implications for Function and Drug Discovery

द्वारा Kojetin, Douglas J., Burris, Thomas P.
प्रकाशित 2013

REV-ERB and ROR nuclear receptors as drug targets

द्वारा Kojetin, Douglas J., Burris, Thomas P.
में प्रकाशित Nat Rev Drug Discov (2014)

The REV-ERBs and RORs: molecular links between circadian rhythms and lipid homeostasis

द्वारा Solt, Laura A, Kojetin, Douglas J, Burris, Thomas P
प्रकाशित 2011

Characterization of the Core Mammalian Clock Component, NPAS2, as a REV-ERBα/RORα Target Gene

द्वारा Crumbley, Christine, Wang, Yongjun, Kojetin, Douglas J., Burris, Thomas P.
प्रकाशित 2010

Activity-based profiling reveals a regulatory link between oxidative stress and protein arginine phosphorylation

द्वारा Fuhrmann, Jakob, Subramanian, Venkataraman, Kojetin, Douglas J., Thompson, Paul R.
में प्रकाशित Cell Chem Biol (2016)

(1)H, (13)C and (15)N chemical shift assignments for the human Pitx2 homeodomain and a R24H homeodomain mutant

द्वारा Doerdelmann, Thomas, Kojetin, Douglas J., Baird-Titus, Jamie M., Rance, Mark
प्रकाशित 2010

(1)H, (13)C and (15)N chemical shift assignments for the human Pitx2 homeodomain in complex with a 22-base hairpin DNA

द्वारा Doerdelmann, Thomas, Kojetin, Douglas J., Baird-Titus, Jamie M., Rance, Mark
प्रकाशित 2011

Regulation of p53 Stability and Apoptosis by a ROR Agonist

द्वारा Wang, Yongjun, Solt, Laura A., Kojetin, Douglas J., Burris, Thomas P.
प्रकाशित 2012

Alternative Splicing of a β(4) Subunit Proline-Rich Motif Regulates Voltage-Dependent Gating and Toxin Block of Ca(v)2.1 Ca(2+) Channels

द्वारा Helton, Thomas D., Kojetin, Douglas J., Cavanagh, John, Horne, William A.
में प्रकाशित J Neurosci (2002)

Deconvolution of Complex 1D NMR Spectra Using Objective Model Selection

द्वारा Hughes, Travis S., Wilson, Henry D., de Vera, Ian Mitchelle S., Kojetin, Douglas J.
में प्रकाशित PLoS One (2015)

Quantitative structural assessment of graded receptor agonism

द्वारा Shang, Jinsai, Brust, Richard, Griffin, Patrick R., Kamenecka, Theodore M., Kojetin, Douglas J.
में प्रकाशित Proc Natl Acad Sci U S A (2019)

Modification of the Orthosteric PPARγ Covalent Antagonist Scaffold Yields an Improved Dual-Site Allosteric Inhibitor

द्वारा Brust, Richard, Lin, Hua, Fuhrmann, Jakob, Asteian, Alice, Kamenecka, Theodore M., Kojetin, Douglas J.
में प्रकाशित ACS Chem Biol (2017)

Structural and Biophysical Insights into the Ligand-Free Pitx2 Homeodomain and a Ring Dermoid of the Cornea Inducing Homeodomain Mutant

द्वारा Doerdelmann, Thomas, Kojetin, Douglas J., Baird-Titus, Jamie M., Solt, Laura A., Burris, Thomas P., Rance, Mark
प्रकाशित 2012

Assessment of NR4A Ligands that Directly Bind and Modulate the Orphan Nuclear Receptor Nurr1

द्वारा Munoz-Tello, Paola, Lin, Hua, Khan, Pasha, de Vera, Ian Mitchelle S., Kamenecka, Theodore M., Kojetin, Douglas J.
में प्रकाशित J Med Chem (2020)

Structural and motional contributions of the Bacillus subtilis ClpC N-domain in adaptor protein interactions

द्वारा Kojetin, Douglas J., McLaughlin, Patrick D., Thompson, Richele J., Dubnau, David, Prepiak, Peter, Rance, Mark, Cavanagh, John
प्रकाशित 2009

Observing selected domains in multi-domain proteins via sortase-mediated ligation and NMR spectroscopy

द्वारा Refaei, Mary Anne, Combs, Al, Kojetin, Douglas J., Cavanagh, John, Caperelli, Carol, Rance, Mark, Sapitro, Jennifer, Tsang, Pearl
प्रकाशित 2010

Structure of REV-ERBβ Ligand-binding Domain Bound to a Porphyrin Antagonist

द्वारा Matta-Camacho, Edna, Banerjee, Subhashis, Hughes, Travis S., Solt, Laura A., Wang, Yongjun, Burris, Thomas P., Kojetin, Douglas J.
प्रकाशित 2014

Insights into the nature of DNA binding of AbrB-like transcription factors

द्वारा Sullivan, Daniel M., Bobay, Benjamin G., Kojetin, Douglas J., Thompson, Richele J., Rance, Mark, Strauch, Mark A., Cavanagh, John
प्रकाशित 2008

Structural basis of altered potency and efficacy displayed by a major in vivo metabolite of the anti-diabetic PPARγ drug pioglitazone

द्वारा Mosure, Sarah A., Shang, Jinsai, Eberhardt, Jerome, Brust, Richard, Zheng, Jie, Griffin, Patrick R., Forli, Stefano, Kojetin, Douglas J.
में प्रकाशित J Med Chem (2019)

Structural basis for heme-dependent NCoR binding to the transcriptional repressor REV-ERBβ

द्वारा Mosure, Sarah A., Strutzenberg, Timothy S., Shang, Jinsai, Munoz-Tello, Paola, Solt, Laura A., Griffin, Patrick R., Kojetin, Douglas J.
में प्रकाशित Sci Adv (2021)