Demonstration of AutoDock as an Educational Tool for Drug Discovery

por Helgren, Travis R., Hagen, Timothy J.
Publicado en J Chem Educ (2017)

(Z)-4-Chloro-N-{3-[(4-chlorophenyl)sulfonyl]-2,3-dihydrobenzo[d]thiazol-2-ylidene}benzene-sulfonamide

por Watkins, Sydney M., Hagen, Timothy J., Perkins, Timothy S., Zheng, Chong
Publicado en IUCrdata (2017)

Advances in Bacterial Methionine Aminopeptidase Inhibition

por Helgren, Travis R., Wangtrakuldee, Phumvadee, Staker, Bart L., Hagen, Timothy J.
Publicado en Curr Top Med Chem (2016)

Discovery of triazines as selective PDE4B versus PDE4D inhibitors

por Hagen, Timothy J., Mo, Xuesheng, Burgin, Alex B., Fox, David, Zhang, Zheng, Gurney, Mark E.
Publicado 2014

The Identification of Inhibitory Compounds of Rickettsia prowazekii Methionine Aminopeptidase for Antibacterial Applications

por Helgren, Travis R., Seven, Elif S., Chen, Congling, Edwards, Thomas E., Staker, Bart L., Abendroth, Jan, Myler, Peter J., Horn, James R., Hagen, Timothy J.
Publicado en Bioorg Med Chem Lett (2018)

Antibacterial activity of 2-amino-4-hydroxypyrimidine-5-carboxylates and binding to Burkholderia pseudomallei 2-C-methyl-D-erythritol-2,4-cyclodiphosphate synthase

por Watkins, Sydney M., Ghose, Debarati, Blain, Joy M., Grote, Dakota L., Luan, Chi-Hao, Clare, Michael, Meganathan, R., Horn, James R., Hagen, Timothy J.
Publicado en Bioorg Med Chem Lett (2019)

Synthesis and biological evaluation of pyrazolopyrimidines as potential antibacterial agents

por Goshu, Gashaw M., Ghose, Debarati, Bain, Joy M., Pierce, Phillip G., Begley, Darren W., Hewitt, Stephen N., Udell, Hannah S., Myler, Peter J., Meganathan, R, Hagen, Timothy J.
Publicado en Bioorg Med Chem Lett (2015)

Discovery of Inhibitors of Burkholderia pseudomallei Methionine Aminopeptidase with Antibacterial Activity

por Wangtrakuldee, Phumvadee, Byrd, Matthew S., Campos, Cristine G., Henderson, Michael W., Zhang, Zheng, Clare, Michael, Masoudi, Ali, Myler, Peter J., Horn, James R., Cotter, Peggy A., Hagen, Timothy J.
Publicado 2013

Rickettsia prowazekii Methionine Aminopeptidase as a Promising Target for the Development of Antibacterial Agents

por Helgren, Travis R., Chen, Congling, Wangtrakuldee, Phumvadee, Edwards, Thomas E., Staker, Bart L., Abendroth, Jan, Sankaran, Banumathi, Housley, Nicole A., Myler, Peter J., Audia, Jonathon P., Horn, James R., Hagen, Timothy J.
Publicado en Bioorg Med Chem (2016)

Cytidine derivatives as IspF inhibitors of Burkolderia pseudomallei

por Zhang, Zheng, Jakkaraju, Sriram, Blain, Joy, Gogol, Kenneth, Zhao, Lei, Hartley, Robert C., Karlsson, Courtney A., Staker, Bart L., Stewart, Lance J., Myler, Peter J., Clare, Michael, Begley, Darren W., Horn, James R., Hagen, Timothy J
Publicado 2013

Design and Synthesis of Selective Phosphodiesterase 4D (PDE4D) Allosteric Inhibitors for the Treatment of Fragile X Syndrome and Other Brain Disorders

por Gurney, Mark E., Nugent, Richard A., Mo, Xuesheng, Sindac, Janice A., Hagen, Timothy J., Fox, David, O’Donnell, James M., Zhang, Chong, Xu, Ying, Zhang, Han-Ting, Groppi, Vincent E., Bailie, Marc, White, Ronald E., Romero, Donna L., Vellekoop, A. Samuel, Walker, Joel R., Surman, Matthew D., Zhu, Lei, Campbell, Robert F.
Publicado en J Med Chem (2019)