Beyond radio-displacement techniques for Identification of CB(1) Ligands: The First Application of a Fluorescence-quenching Assay

por Bruno, Agostino, Lembo, Francesca, Novellino, Ettore, Stornaiuolo, Mariano, Marinelli, Luciana
Publicado 2014

Membrane-Sensitive Conformational States of Helix 8 in the Metabotropic Glu2 Receptor, a Class C GPCR

por Bruno, Agostino, Costantino, Gabriele, de Fabritiis, Gianni, Pastor, Manuel, Selent, Jana
Publicado 2012

Correction: Membrane-Sensitive Conformational States of Helix 8 in the Metabotropic Glu2 Receptor, a Class C GPCR

por Bruno, Agostino, Costantino, Gabriele, de Fabritiis, Gianni, Pastor, Manuel, Selent, Jana
Publicado 2012

The Glycan Role in the Glycopeptide Immunogenicity Revealed by Atomistic Simulations and Spectroscopic Experiments on the Multiple Sclerosis Biomarker CSF114(Glc)

por Bruno, Agostino, Scrima, Mario, Novellino, Ettore, D'Errico, Gerardino, D'Ursi, Anna Maria, Limongelli, Vittorio
Publicado en Sci Rep (2015)

Endogenous vs Exogenous Allosteric Modulators in GPCRs: A dispute for shuttling CB(1) among different membrane microenvironments

por Stornaiuolo, Mariano, Bruno, Agostino, Botta, Lorenzo, Regina, Giuseppe La, Cosconati, Sandro, Silvestri, Romano, Marinelli, Luciana, Novellino, Ettore
Publicado en Sci Rep (2015)

Biochemical Characterization of Aspergillus fumigatus AroH, a Putative Aromatic Amino Acid Aminotransferase

por Dindo, Mirco, Costanzi, Egidia, Pieroni, Marco, Costantini, Claudio, Annunziato, Giannamaria, Bruno, Agostino, Keller, Nancy P., Romani, Luigina, Zelante, Teresa, Cellini, Barbara
Publicado en Front Mol Biosci (2018)

Inhibition of Nonessential Bacterial Targets: Discovery of a Novel Serine O-Acetyltransferase Inhibitor

por Magalhães, Joana, Franko, Nina, Raboni, Samanta, Annunziato, Giannamaria, Tammela, Päivi, Bruno, Agostino, Bettati, Stefano, Mozzarelli, Andrea, Pieroni, Marco, Campanini, Barbara, Costantino, Gabriele
Publicado en ACS Med Chem Lett (2020)

Discovery of novel fragments inhibiting O-acetylserine sulphhydrylase by combining scaffold hopping and ligand–based drug design

por Magalhães, Joana, Franko, Nina, Annunziato, Giannamaria, Welch, Martin, Dolan, Stephen K., Bruno, Agostino, Mozzarelli, Andrea, Armao, Stefano, Jirgensons, Aigars, Pieroni, Marco, Costantino, Gabriele, Campanini, Barbara
Publicado en J Enzyme Inhib Med Chem (2018)

Discovering a new class of antifungal agents that selectively inhibits microbial carbonic anhydrases

por Annunziato, Giannamaria, Giovati, Laura, Angeli, Andrea, Pavone, Marialaura, Del Prete, Sonia, Pieroni, Marco, Capasso, Clemente, Bruno, Agostino, Conti, Stefania, Magliani, Walter, Supuran, Claudiu T., Costantino, Gabriele
Publicado en J Enzyme Inhib Med Chem (2018)

Discovery of Substituted (2-Aminooxazol-4-yl)Isoxazole-3-carboxylic Acids as Inhibitors of Bacterial Serine Acetyltransferase in the Quest for Novel Potential Antibacterial Adjuvan...

por Magalhães, Joana, Franko, Nina, Raboni, Samanta, Annunziato, Giannamaria, Tammela, Päivi, Bruno, Agostino, Bettati, Stefano, Armao, Stefano, Spadini, Costanza, Cabassi, Clotilde Silvia, Mozzarelli, Andrea, Pieroni, Marco, Campanini, Barbara, Costantino, Gabriele
Publicado en Pharmaceuticals (Basel) (2021)

The Aryl Hydrocarbon Receptor (AhR) Mediates the Counter-Regulatory Effects of Pelargonidins in Models of Inflammation and Metabolic Dysfunctions

por Biagioli, Michele, Carino, Adriana, Fiorucci, Chiara, Annunziato, Giannamaria, Marchianò, Silvia, Bordoni, Martina, Roselli, Rosalinda, Giorgio, Cristina Di, Castiglione, Federica, Ricci, Patrizia, Bruno, Agostino, Faccini, Andrea, Distrutti, Eleonora, Baldoni, Monia, Costantino, Gabriele, Fiorucci, Stefano
Publicado en Nutrients (2019)

Molecular mechanism and functional role of brefeldin A-mediated ADP-ribosylation of CtBP1/BARS

por Colanzi, Antonino, Grimaldi, Giovanna, Catara, Giuliana, Valente, Carmen, Cericola, Claudia, Liberali, Prisca, Ronci, Maurizio, Lalioti, Vasiliki S., Bruno, Agostino, Beccari, Andrea R., Urbani, Andrea, De Flora, Antonio, Nardini, Marco, Bolognesi, Martino, Luini, Alberto, Corda, Daniela
Publicado 2013

Binding of the Anti-FIV Peptide C8 to Differently Charged Membrane Models: From First Docking to Membrane Tubulation

por Di Marino, Daniele, Bruno, Agostino, Grimaldi, Manuela, Scrima, Mario, Stillitano, Ilaria, Amodio, Giuseppina, Della Sala, Grazia, Romagnoli, Alice, De Santis, Augusta, Moltedo, Ornella, Remondelli, Paolo, Boccia, Giovanni, D'Errico, Gerardino, D'Ursi, Anna Maria, Limongelli, Vittorio
Publicado en Front Chem (2020)

Everolimus induces Met inactivation by disrupting the FKBP12/Met complex

por Raimondo, Lucia, D'Amato, Valentina, Servetto, Alberto, Rosa, Roberta, Marciano, Roberta, Formisano, Luigi, Mauro, Concetta Di, Orsini, Roberta Clara, Cascetta, Priscilla, Ciciola, Paola, De Maio, Ana Paula, Di Renzo, Maria Flavia, Cosconati, Sandro, Bruno, Agostino, Randazzo, Antonio, Napolitano, Filomena, Montuori, Nunzia, Veneziani, Bianca Maria, Placido, Sabino De, Bianco, Roberto
Publicado en Oncotarget (2016)

Targeting the minor pocket of C5aR for the rational design of an oral allosteric inhibitor for inflammatory and neuropathic pain relief

por Moriconi, Alessio, Cunha, Thiago M., Souza, Guilherme R., Lopes, Alexandre H., Cunha, Fernando Q., Carneiro, Victor L., Pinto, Larissa G., Brandolini, Laura, Aramini, Andrea, Bizzarri, Cinzia, Bianchini, Gianluca, Beccari, Andrea R., Fanton, Marco, Bruno, Agostino, Costantino, Gabriele, Bertini, Riccardo, Galliera, Emanuela, Locati, Massimo, Ferreira, Sérgio H., Teixeira, Mauro M., Allegretti, Marcello
Publicado en Proc Natl Acad Sci U S A (2014)