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Chemical features important for activity in a class of inhibitors targeting the Wip1 flap subdomain

The wild-type p53 induced phosphatase 1, Wip1 (PP2Cδ), is a PP2C family Ser/Thr phosphatase that negatively regulates the function of multiple proteins such as p53, ATM, Chk1, Chk2, Mdm2 and p38 MAPK involved in a DNA damage response. Wip1 dephosphorylates and inactivates its protein targets which a...

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Publicat a:ChemMedChem
Autors principals: Tagad, Harichandra D., Debnath, Subrata, Clausse, Victor, Saha, Mrinmoy, Mazur, Sharlyn, Appella, Ettore, Appella, Daniel H.
Format: Artigo
Idioma:Inglês
Publicat: 2018
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC8022280/
https://ncbi.nlm.nih.gov/pubmed/29476592
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/cmdc.201700779
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