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Linker Hydrophilicity Modulates the Anticancer Activity of RGD–Cryptophycin Conjugates

Most anticancer agents are hydrophobic and can easily penetrate the tumor cell membrane by passive diffusion. This may impede the development of highly effective and tumor‐selective treatment options. A hydrophilic β‐glucuronidase‐cleavable linker was used to connect the highly potent antimitotic ag...

Ausführliche Beschreibung

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Bibliographische Detailangaben
Veröffentlicht in:Chemistry
Hauptverfasser: Anselmi, Michele, Borbély, Adina, Figueras, Eduard, Michalek, Carmela, Kemker, Isabell, Gentilucci, Luca, Sewald, Norbert
Format: Artigo
Sprache:Inglês
Veröffentlicht: John Wiley and Sons Inc. 2020
Schlagworte:
Online Zugang:https://ncbi.nlm.nih.gov/pmc/articles/PMC7839693/
https://ncbi.nlm.nih.gov/pubmed/32955139
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/chem.202003471
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