Cargando...

Linker Hydrophilicity Modulates the Anticancer Activity of RGD–Cryptophycin Conjugates

Most anticancer agents are hydrophobic and can easily penetrate the tumor cell membrane by passive diffusion. This may impede the development of highly effective and tumor‐selective treatment options. A hydrophilic β‐glucuronidase‐cleavable linker was used to connect the highly potent antimitotic ag...

Descrición completa

Gardado en:
Detalles Bibliográficos
Publicado en:Chemistry
Main Authors: Anselmi, Michele, Borbély, Adina, Figueras, Eduard, Michalek, Carmela, Kemker, Isabell, Gentilucci, Luca, Sewald, Norbert
Formato: Artigo
Idioma:Inglês
Publicado: John Wiley and Sons Inc. 2020
Assuntos:
Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC7839693/
https://ncbi.nlm.nih.gov/pubmed/32955139
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/chem.202003471
Tags: Engadir etiqueta
Sen Etiquetas, Sexa o primeiro en etiquetar este rexistro!