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Proton-sensing G protein-coupled receptors: detectors of tumor acidosis and candidate drug targets

Cells in tumor microenvironments (TMEs) use several mechanisms to sense their low pH (<7.0), including via proton-sensing G protein-coupled receptors (psGPCRs): GPR4, GPR65/TDAG8, GPR68/OGR1 and GPR132/G2A. Numerous cancers have increased expression of psGPCRs. The psGPCRs may contribute to featu...

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Dettagli Bibliografici
Pubblicato in:Future Med Chem
Autori principali: Insel, Paul A, Sriram, Krishna, Salmerón, Cristina, Wiley, Shu Z
Natura: Artigo
Lingua:Inglês
Pubblicazione: Newlands Press Ltd 2020
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC7607387/
https://ncbi.nlm.nih.gov/pubmed/32116003
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.4155/fmc-2019-0357
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