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Intramolecular vinylation of aryl rings by vinyl cations

A Lewis acid mediated intramolecular electrophilic vinylation of aryl rings by vinyl cations is reported. This reaction takes advantage of β-hydroxy-α-diazo ketones as vinyl cation precursors and provides good yields of tricyclic 1-indenones that contain a 7-membered ring. Extending the alkane chain...

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Publicat a:Org Lett
Autors principals: Fang, Jian, Brewer, Matthias
Format: Artigo
Idioma:Inglês
Publicat: 2018
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC7045802/
https://ncbi.nlm.nih.gov/pubmed/30426753
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.orglett.8b03054
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