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Designing Functionally Selective Noncatechol Dopamine D(1) Receptor Agonists with Potent In Vivo Antiparkinsonian Activity

Dopamine receptors are important G protein-coupled receptors (GPCRs) with therapeutic opportunities for treating Parkinson’s Disease (PD) motor and cognitive deficits. Biased D(1) dopamine ligands that differentially activate G protein over β-arrestin recruitment pathways are valuable chemical tools...

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Detalhes bibliográficos
Publicado no:ACS Chem Neurosci
Main Authors: Martini, Michael L., Ray, Caroline, Yu, Xufen, Liu, Jing, Pogorelov, Vladimir M., Wetsel, William C., Huang, Xi-Ping, McCorvy, John D., Caron, Marc G., Jin, Jian
Formato: Artigo
Idioma:Inglês
Publicado em: 2019
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC6785188/
https://ncbi.nlm.nih.gov/pubmed/31387346
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acschemneuro.9b00410
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