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Improved predictions of time-dependent drug-drug interactions by determination of cytosolic drug concentrations

The clinical impact of drug-drug interactions based on time-dependent inhibition of cytochrome P450 (CYP) 3A4 has often been overpredicted, likely due to use of improper inhibitor concentration estimates at the enzyme. Here, we investigated if use of cytosolic unbound inhibitor concentrations could...

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Bibliographische Detailangaben
Veröffentlicht in:Sci Rep
Hauptverfasser: Filppula, Anne M., Parvizi, Rezvan, Mateus, André, Baranczewski, Pawel, Artursson, Per
Format: Artigo
Sprache:Inglês
Veröffentlicht: Nature Publishing Group UK 2019
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Online Zugang:https://ncbi.nlm.nih.gov/pmc/articles/PMC6458156/
https://ncbi.nlm.nih.gov/pubmed/30971754
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/s41598-019-42051-x
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