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Intracellular drug bioavailability: a new predictor of system dependent drug disposition

Intracellular drug exposure is influenced by cell- and tissue-dependent expression of drug-transporting proteins and metabolizing enzymes. Here, we introduce the concept of intracellular bioavailability (F(ic)) as the fraction of extracellular drug available to bind intracellular targets, and we ass...

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Publicat a:Sci Rep
Autors principals: Mateus, André, Treyer, Andrea, Wegler, Christine, Karlgren, Maria, Matsson, Pär, Artursson, Per
Format: Artigo
Idioma:Inglês
Publicat: Nature Publishing Group 2017
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC5320532/
https://ncbi.nlm.nih.gov/pubmed/28225057
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/srep43047
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