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Impact of Intracellular Concentrations on Metabolic Drug-Drug Interaction Studies

Accurate prediction of drug-drug interactions (DDI) is a challenging task in drug discovery and development. It requires determination of enzyme inhibition in vitro which is highly system-dependent for many compounds. The aim of this study was to investigate whether the determination of intracellula...

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Publicat a:AAPS J
Autors principals: Treyer, Andrea, Ullah, Mohammed, Parrott, Neil, Molitor, Birgit, Fowler, Stephen, Artursson, Per
Format: Artigo
Idioma:Inglês
Publicat: Springer International Publishing 2019
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC6581936/
https://ncbi.nlm.nih.gov/pubmed/31214810
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1208/s12248-019-0344-8
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