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Analysis of equilibrium binding of an orthosteric tracer and two allosteric modulators

Allosteric ligands bind to receptors at sites that are distinct from those endogenous agonists and orthosteric pharmacological agents interact with. Both an allosteric and orthosteric ligand bind simultaneously to the receptor to form a ternary complex, where each ligand influences binding affinity...

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Dades bibliogràfiques
Publicat a:PLoS One
Autors principals: Jakubík, Jan, Randáková, Alena, El-Fakahany, Esam E., Doležal, Vladimír
Format: Artigo
Idioma:Inglês
Publicat: Public Library of Science 2019
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC6436737/
https://ncbi.nlm.nih.gov/pubmed/30917186
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1371/journal.pone.0214255
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