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Divergence of allosteric effects of rapacuronium on binding and function of muscarinic receptors

BACKGROUND: Many neuromuscular blockers act as negative allosteric modulators of muscarinic acetylcholine receptors by decreasing affinity and potency of acetylcholine. The neuromuscular blocker rapacuronium has been shown to have facilitatory effects at muscarinic receptors leading to bronchospasm....

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Autori principali: Jakubík, Jan, Randáková, Alena, El-Fakahany, Esam E, Doležal, Vladimír
Natura: Artigo
Lingua:Inglês
Pubblicazione: BioMed Central 2009
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC2806265/
https://ncbi.nlm.nih.gov/pubmed/20038295
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1186/1471-2210-9-15
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