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Analysis of equilibrium binding of an orthosteric tracer and two allosteric modulators

Allosteric ligands bind to receptors at sites that are distinct from those endogenous agonists and orthosteric pharmacological agents interact with. Both an allosteric and orthosteric ligand bind simultaneously to the receptor to form a ternary complex, where each ligand influences binding affinity...

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Detalles Bibliográficos
Publicado en:PLoS One
Main Authors: Jakubík, Jan, Randáková, Alena, El-Fakahany, Esam E., Doležal, Vladimír
Formato: Artigo
Idioma:Inglês
Publicado: Public Library of Science 2019
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC6436737/
https://ncbi.nlm.nih.gov/pubmed/30917186
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1371/journal.pone.0214255
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