Llwytho...

Analysis of equilibrium binding of an orthosteric tracer and two allosteric modulators

Allosteric ligands bind to receptors at sites that are distinct from those endogenous agonists and orthosteric pharmacological agents interact with. Both an allosteric and orthosteric ligand bind simultaneously to the receptor to form a ternary complex, where each ligand influences binding affinity...

Disgrifiad llawn

Wedi'i Gadw mewn:
Manylion Llyfryddiaeth
Cyhoeddwyd yn:PLoS One
Prif Awduron: Jakubík, Jan, Randáková, Alena, El-Fakahany, Esam E., Doležal, Vladimír
Fformat: Artigo
Iaith:Inglês
Cyhoeddwyd: Public Library of Science 2019
Pynciau:
Mynediad Ar-lein:https://ncbi.nlm.nih.gov/pmc/articles/PMC6436737/
https://ncbi.nlm.nih.gov/pubmed/30917186
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1371/journal.pone.0214255
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