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The operational model of allosteric modulation of pharmacological agonism

Proper determination of agonist efficacy is indispensable in the evaluation of agonist selectivity and bias to activation of specific signalling pathways. The operational model (OM) of pharmacological agonism is a useful means for achieving this goal. Allosteric ligands bind to receptors at sites th...

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Detalles Bibliográficos
Publicado en:Sci Rep
Main Authors: Jakubík, Jan, Randáková, Alena, Chetverikov, Nikolai, El-Fakahany, Esam E., Doležal, Vladimír
Formato: Artigo
Idioma:Inglês
Publicado: Nature Publishing Group UK 2020
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC7468285/
https://ncbi.nlm.nih.gov/pubmed/32879329
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/s41598-020-71228-y
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