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Structure-Guided Modification of Heterocyclic Antagonists of the P2Y(14) Receptor

The P2Y(14) receptor (P2Y(14)R) mediates inflammatory activity by activating neutrophil motility, but few classes of antagonists are known. We have explored the structure activity relationship of a 3-(4-phenyl- 1H-1,2,3-triazol-1-yl)-5-(aryl)benzoic acid antagonist scaffold, assisted by docking and...

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Bibliographische Detailangaben
Veröffentlicht in:J Med Chem
Hauptverfasser: Yu, Jinha, Ciancetta, Antonella, Dudas, Steven, Duca, Sierra, Lottermoser, Justine, Jacobson, Kenneth A.
Format: Artigo
Sprache:Inglês
Veröffentlicht: 2018
Schlagworte:
Online Zugang:https://ncbi.nlm.nih.gov/pmc/articles/PMC6428052/
https://ncbi.nlm.nih.gov/pubmed/29767967
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.jmedchem.8b00168
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