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Structure-Guided Modification of Heterocyclic Antagonists of the P2Y(14) Receptor

The P2Y(14) receptor (P2Y(14)R) mediates inflammatory activity by activating neutrophil motility, but few classes of antagonists are known. We have explored the structure activity relationship of a 3-(4-phenyl- 1H-1,2,3-triazol-1-yl)-5-(aryl)benzoic acid antagonist scaffold, assisted by docking and...

Täydet tiedot

Tallennettuna:
Bibliografiset tiedot
Julkaisussa:J Med Chem
Päätekijät: Yu, Jinha, Ciancetta, Antonella, Dudas, Steven, Duca, Sierra, Lottermoser, Justine, Jacobson, Kenneth A.
Aineistotyyppi: Artigo
Kieli:Inglês
Julkaistu: 2018
Aiheet:
Linkit:https://ncbi.nlm.nih.gov/pmc/articles/PMC6428052/
https://ncbi.nlm.nih.gov/pubmed/29767967
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.jmedchem.8b00168
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