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Fenestrations control resting-state block of a voltage-gated sodium channel

Potency of drug action is usually determined by binding to a specific receptor site on target proteins. In contrast to this conventional paradigm, we show here that potency of local anesthetics (LAs) and antiarrhythmic drugs (AADs) that block sodium channels is controlled by fenestrations that allow...

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Detalhes bibliográficos
Publicado no:Proc Natl Acad Sci U S A
Main Authors: Gamal El-Din, Tamer M., Lenaeus, Michael J., Zheng, Ning, Catterall, William A.
Formato: Artigo
Idioma:Inglês
Publicado em: National Academy of Sciences 2018
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC6304959/
https://ncbi.nlm.nih.gov/pubmed/30518562
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1073/pnas.1814928115
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