Carregant...

Fenestrations control resting-state block of a voltage-gated sodium channel

Potency of drug action is usually determined by binding to a specific receptor site on target proteins. In contrast to this conventional paradigm, we show here that potency of local anesthetics (LAs) and antiarrhythmic drugs (AADs) that block sodium channels is controlled by fenestrations that allow...

Descripció completa

Guardat en:
Dades bibliogràfiques
Publicat a:Proc Natl Acad Sci U S A
Autors principals: Gamal El-Din, Tamer M., Lenaeus, Michael J., Zheng, Ning, Catterall, William A.
Format: Artigo
Idioma:Inglês
Publicat: National Academy of Sciences 2018
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC6304959/
https://ncbi.nlm.nih.gov/pubmed/30518562
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1073/pnas.1814928115
Etiquetes: Afegir etiqueta
Sense etiquetes, Sigues el primer a etiquetar aquest registre!