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Fenestrations control resting-state block of a voltage-gated sodium channel

Potency of drug action is usually determined by binding to a specific receptor site on target proteins. In contrast to this conventional paradigm, we show here that potency of local anesthetics (LAs) and antiarrhythmic drugs (AADs) that block sodium channels is controlled by fenestrations that allow...

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Bibliografski detalji
Izdano u:Proc Natl Acad Sci U S A
Glavni autori: Gamal El-Din, Tamer M., Lenaeus, Michael J., Zheng, Ning, Catterall, William A.
Format: Artigo
Jezik:Inglês
Izdano: National Academy of Sciences 2018
Teme:
Online pristup:https://ncbi.nlm.nih.gov/pmc/articles/PMC6304959/
https://ncbi.nlm.nih.gov/pubmed/30518562
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1073/pnas.1814928115
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