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Identifying Functional Hotspot Residues for Biased Ligand Design in G-Protein-Coupled Receptors

G-protein-coupled receptors (GPCRs) mediate multiple signaling pathways in the cell, depending on the agonist that activates the receptor and multiple cellular factors. Agonists that show higher potency to specific signaling pathways over others are known as “biased agonists” and have been shown to...

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Библиографические подробности
Опубликовано в: :Mol Pharmacol
Главные авторы: Nivedha, Anita K., Tautermann, Christofer S., Bhattacharya, Supriyo, Lee, Sangbae, Casarosa, Paola, Kollak, Ines, Kiechle, Tobias, Vaidehi, Nagarajan
Формат: Artigo
Язык:Inglês
Опубликовано: The American Society for Pharmacology and Experimental Therapeutics 2018
Предметы:
Online-ссылка:https://ncbi.nlm.nih.gov/pmc/articles/PMC5832328/
https://ncbi.nlm.nih.gov/pubmed/29367258
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/mol.117.110395
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