Metabolic Profiling of CB1 Neutral Antagonists

PIMSR is among the first neutral antagonists for the CB1R and was demonstrated pharmacologically to bind to the CB1R, yet not alter calcium flux. It was further shown computationally to be able to stabilize both the active and inactive states of CB1R revealing the molecular interactions that mechani...

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Bibliografiske detaljer
Udgivet i:Methods Enzymol
Main Authors: Seltzman, Herbert H., Maitra, Rangan, Bortoff, Katharine, Henson, Jay, Reggio, Patricia H., Wesley, Daniel, Tam, Joseph
Format: Artigo
Sprog:Inglês
Udgivet: 2017
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Article
Online adgang:https://ncbi.nlm.nih.gov/pmc/articles/PMC5802864/
https://ncbi.nlm.nih.gov/pubmed/28750803
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/bs.mie.2017.06.025
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