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Towards rational design of cannabinoid receptor 1 (CB1) antagonists for peripheral selectivity

CB1 receptor antagonists that are peripherally restricted were targeted. Compounds with permanent charge as well as compounds that have increased polar surface area were made and tested against CB1 for binding and activity. Sulfonamide and sulfamide with high polar surface area and good activity at...

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Detalhes bibliográficos
Main Authors: Fulp, Alan, Bortoff, Katherine, Zhang, Yanan, Seltzman, Herbert, Snyder, Rodney, Maitra, Rangan
Formato: Artigo
Idioma:Inglês
Publicado em: 2011
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC3171605/
https://ncbi.nlm.nih.gov/pubmed/21875798
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmcl.2011.08.032
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