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Synthesis of sulfamoylbenzamide derivatives as HBV capsid assembly effector
The synthesis of novel series of sulfamoylbenzamides as HBV capsid assembly effector is reported. The structure was divided into five parts which were independently modified as part of our lead optimization. All synthesized compounds were evaluated for their anti-HBV activity and toxicity in human h...
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| Опубликовано в: : | Eur J Med Chem |
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| Главные авторы: | , , , , , , , |
| Формат: | Artigo |
| Язык: | Inglês |
| Опубликовано: |
2017
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| Предметы: | |
| Online-ссылка: | https://ncbi.nlm.nih.gov/pmc/articles/PMC5581232/ https://ncbi.nlm.nih.gov/pubmed/28688280 https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.ejmech.2017.06.062 |
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