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Engineering Pak1 allosteric switches

p21-activated kinases (PAKs) are important regulators of cell motility and morphology. It has been challenging to interrogate their functions because cells adapt to genetic manipulation of PAK, and because inhibitors act on multiple PAK isoforms. Here we describe genetically encoded PAK1 analogues t...

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Publicat a:ACS Synth Biol
Autors principals: Dagliyan, Onur, Karginov, Andrei V., Yagishita, Sho, Gale, Madeline E., Wang, Hui, DerMardirossian, Celine, Wells, Claire M., Dokholyan, Nikolay V., Kasai, Haruo, Hahn, Klaus M.
Format: Artigo
Idioma:Inglês
Publicat: 2017
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC5562282/
https://ncbi.nlm.nih.gov/pubmed/28365983
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acssynbio.6b00359
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