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Development of a potent 2-oxoamide inhibitor of secreted phospholipase A(2) guided by molecular docking calculations and molecular dynamics simulations

Inhibition of group IIA secreted phospholipase A(2) (GIIA sPLA(2)) has been an important objective for medicinal chemists. We have previously shown that inhibitors incorporating the 2-oxoamide functionality may inhibit human and mouse GIIA sPLA(2)s. Herein, the development of new potent inhibitors b...

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Detalhes bibliográficos
Publicado no:Bioorg Med Chem
Main Authors: Vasilakaki, Sofia, Barbayianni, Efrosini, Leonis, Georgios, Papadopoulos, Manthos G., Mavromoustakos, Thomas, Gelb, Michael H., Kokotos, George
Formato: Artigo
Idioma:Inglês
Publicado em: 2016
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC5292099/
https://ncbi.nlm.nih.gov/pubmed/26970660
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmc.2016.02.040
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