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Protein disulfide isomerase inhibition blocks thrombin generation in humans by interfering with platelet factor V activation

BACKGROUND: Protein disulfide isomerase (PDI) is required for thrombus formation. We previously demonstrated that glycosylated quercetin flavonoids such as isoquercetin inhibit PDI activity and thrombus formation in animal models, but whether extracellular PDI represents a viable anticoagulant targe...

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Foilsithe in:JCI Insight
Main Authors: Stopa, Jack D., Neuberg, Donna, Puligandla, Maneka, Furie, Bruce, Flaumenhaft, Robert, Zwicker, Jeffrey I.
Formáid: Artigo
Teanga:Inglês
Foilsithe: American Society for Clinical Investigation 2017
Ábhair:
Rochtain Ar Líne:https://ncbi.nlm.nih.gov/pmc/articles/PMC5214567/
https://ncbi.nlm.nih.gov/pubmed/28097231
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1172/jci.insight.89373
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