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Protein disulfide isomerase inhibition blocks thrombin generation in humans by interfering with platelet factor V activation

BACKGROUND: Protein disulfide isomerase (PDI) is required for thrombus formation. We previously demonstrated that glycosylated quercetin flavonoids such as isoquercetin inhibit PDI activity and thrombus formation in animal models, but whether extracellular PDI represents a viable anticoagulant targe...

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Publicado en:JCI Insight
Autores principales: Stopa, Jack D., Neuberg, Donna, Puligandla, Maneka, Furie, Bruce, Flaumenhaft, Robert, Zwicker, Jeffrey I.
Formato: Artigo
Lenguaje:Inglês
Publicado: American Society for Clinical Investigation 2017
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC5214567/
https://ncbi.nlm.nih.gov/pubmed/28097231
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1172/jci.insight.89373
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