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Decreasing Distortion Energies without Strain: Diazo-Selective 1,3-Dipolar Cycloadditions

The diazo group has attributes that complement those of the azido group for applications in chemical biology. Here, we use computational analyses to provide insights into the chemoselectivity of the diazo group in 1,3-dipolar cycloadditions. Dipole distortion energies are responsible for ~80% of the...

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Pubblicato in:J Org Chem
Autori principali: Gold, Brian, Aronoff, Matthew R., Raines, Ronald T.
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2016
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC5141247/
https://ncbi.nlm.nih.gov/pubmed/27332711
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.joc.6b00948
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