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Structure, Function and Inhibition of Staphylococcus aureus Heptaprenyl Diphosphate Synthase

We report the first structure of heptaprenyl diphosphate synthase from Staphylococcus aureus (SaHepPPS), together with an investigation of its mechanism of action, and inhibition. The protein is involved in the formation of menaquinone, a key electron transporter in many bacteria, including pathogen...

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Dades bibliogràfiques
Publicat a:ChemMedChem
Autors principals: Desai, Janish, Liu, Yi-Liang, Wei, Hongli, Liu, Weidong, Ko, Tzu-Ping, Guo, Rey-Ting, Oldfield, Eric
Format: Artigo
Idioma:Inglês
Publicat: 2016
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC5012948/
https://ncbi.nlm.nih.gov/pubmed/27457559
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/cmdc.201600311
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