A carregar...

Interactions between amiodarone and the hERG potassium channel pore determined with mutagenesis and in silico docking

The antiarrhythmic drug amiodarone delays cardiac repolarisation through inhibition of hERG-encoded potassium channels responsible for the rapid delayed rectifier potassium current (I(Kr)). This study aimed to elucidate molecular determinants of amiodarone binding to the hERG channel. Whole-cell pat...

ver descrição completa

Na minha lista:
Detalhes bibliográficos
Publicado no:Biochem Pharmacol
Main Authors: Zhang, Yihong, Colenso, Charlotte K., El Harchi, Aziza, Cheng, Hongwei, Witchel, Harry J., Dempsey, Chris E., Hancox, Jules C.
Formato: Artigo
Idioma:Inglês
Publicado em: Elsevier Science 2016
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC4959829/
https://ncbi.nlm.nih.gov/pubmed/27256139
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bcp.2016.05.013
Tags: Adicionar Tag
Sem tags, seja o primeiro a adicionar uma tag!