Caricamento...

The Investigational Drug VT-1129 Is a Highly Potent Inhibitor of Cryptococcus Species CYP51 but Only Weakly Inhibits the Human Enzyme

Cryptococcosis is a life-threatening disease often associated with HIV infection. Three Cryptococcus species CYP51 enzymes were purified and catalyzed the 14α-demethylation of lanosterol, eburicol, and obtusifoliol. The investigational agent VT-1129 bound tightly to all three CYP51 proteins (dissoci...

Descrizione completa

Salvato in:
Dettagli Bibliografici
Pubblicato in:Antimicrob Agents Chemother
Autori principali: Warrilow, Andrew G. S., Parker, Josie E., Price, Claire L., Nes, W. David, Garvey, Edward P., Hoekstra, William J., Schotzinger, Robert J., Kelly, Diane E., Kelly, Steven L.
Natura: Artigo
Lingua:Inglês
Pubblicazione: American Society for Microbiology 2016
Soggetti:
Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC4958158/
https://ncbi.nlm.nih.gov/pubmed/27161631
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1128/AAC.00349-16
Tags: Aggiungi Tag
Nessun Tag, puoi essere il primo ad aggiungerne! !