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Bromopyridone Nucleotide Analogues, Anoxic Selective Radiosensitizing Agents That Are Incorporated in DNA by Polymerases

Ionizing radiation is frequently used to kill tumor cells. However, hypoxic solid tumor cells are more resistant to this treatment, providing the impetus to develop molecules that sensitize cells to ionizing radiation. 5-Bromo-2′-deoxyuridine (BrdU) has been investigated as a radiosensitizing agent...

Πλήρης περιγραφή

Αποθηκεύτηκε σε:
Λεπτομέρειες βιβλιογραφικής εγγραφής
Τόπος έκδοσης:J Org Chem
Κύριοι συγγραφείς: Rudra, Arnab, Hou, Dianjie, Zhang, Yonggang, Coulter, Jonathan, Zhou, Haoming, DeWeese, Theodore L., Greenberg, Marc M.
Μορφή: Artigo
Γλώσσα:Inglês
Έκδοση: 2015
Θέματα:
Διαθέσιμο Online:https://ncbi.nlm.nih.gov/pmc/articles/PMC4877698/
https://ncbi.nlm.nih.gov/pubmed/26509218
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.joc.5b01833
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