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Evaluation of TK1 targeting carboranyl thymidine analogues as potential delivery agents for neutron capture therapy of brain tumors

In this report we describe studies with N5-2OH, a carboranyl thymidine analogue (CTA) that is a substrate for thymidine kinase 1 (TK1), using the F98 rat glioma model. In vivo BNCT studies have demonstrated that intracerebral (i.c.) osmotic pump infusion of N5-2OH yielded survival data equivalent to...

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Publicat a:Appl Radiat Isot
Autors principals: Barth, Rolf F., Yang, Weilian, Nakkula, Robin J., Byun, Youngjoo, Tjarks, Werner, Wu, Lai Chu, Binns, Peter J., Riley, Kent J.
Format: Artigo
Idioma:Inglês
Publicat: 2015
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC4685942/
https://ncbi.nlm.nih.gov/pubmed/26282567
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.apradiso.2015.06.031
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