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Blockade of non-opioid excitatory effects of spinal dynorphin A at bradykinin receptors

Dynorphin A (Dyn A) is an endogenous opioid ligand that possesses neuroinhibitory (antinociceptive) effects via μ, δ, and κ opioid receptors. However, under chronic pain conditions, up-regulated spinal Dyn A can also interact with bradykinin receptors (BRs) to promote hyperalgesia through a neuroexc...

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Detalhes bibliográficos
Publicado no:Receptors Clin Investig
Main Authors: Lee, Yeon Sun, Hall, Sara M., Ramos-Colon, Cyf, Remesic, Michael, Rankin, David, Vanderah, Todd W., Porreca, Frank, Lai, Josephine, Hruby, Victor J.
Formato: Artigo
Idioma:Inglês
Publicado em: 2015
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC4515361/
https://ncbi.nlm.nih.gov/pubmed/26221618
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.14800/rci.517
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