Učitavanje...

A bump-and-hole approach to engineer controlled selectivity of BET bromodomain chemical probes

Small molecules are useful tools for probing the biological function and therapeutic potential of individual proteins, but achieving selectivity is challenging when the target protein shares structural domains with other proteins. The Bromo and Extra-Terminal (BET) proteins have attracted interest b...

Cijeli opis

Spremljeno u:
Bibliografski detalji
Izdano u:Science
Glavni autori: Baud, Matthias G. J., Lin-Shiao, Enrique, Cardote, Teresa, Tallant, Cynthia, Pschibul, Annica, Chan, Kwok-Ho, Zengerle, Michael, Garcia, Jordi R., Kwan, Terence T.-L., Ferguson, Fleur M., Ciulli, Alessio
Format: Artigo
Jezik:Inglês
Izdano: 2014
Teme:
Online pristup:https://ncbi.nlm.nih.gov/pmc/articles/PMC4458378/
https://ncbi.nlm.nih.gov/pubmed/25323695
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1126/science.1249830
Oznake: Dodaj oznaku
Bez oznaka, Budi prvi tko označuje ovaj zapis!