New Synthetic Routes to Triazolo-benzodiazepine Analogues: Expanding the Scope of the Bump-and-Hole Approach for Selective Bromo and Extra-Terminal (BET) Bromodomain Inhibition

Por Baud, Matthias G. J., Lin-Shiao, Enrique, Zengerle, Michael, Tallant, Cynthia, Ciulli, Alessio
Publicado no J Med Chem (2015)

Comprehensive analysis of histone post-translational modifications in mouse and human male germ cells

Por Luense, Lacey J., Wang, Xiaoshi, Schon, Samantha B., Weller, Angela H., Lin Shiao, Enrique, Bryant, Jessica M., Bartolomei, Marisa S., Coutifaris, Christos, Garcia, Benjamin A., Berger, Shelley L.
Publicado no Epigenetics Chromatin (2016)

A bump-and-hole approach to engineer controlled selectivity of BET bromodomain chemical probes

Por Baud, Matthias G. J., Lin-Shiao, Enrique, Cardote, Teresa, Tallant, Cynthia, Pschibul, Annica, Chan, Kwok-Ho, Zengerle, Michael, Garcia, Jordi R., Kwan, Terence T.-L., Ferguson, Fleur M., Ciulli, Alessio
Publicado no Science (2014)