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Stabilization of G protein-coupled receptors by point mutations

G protein-coupled receptors (GPCRs) are flexible integral membrane proteins involved in transmembrane signaling. Their involvement in many physiological processes makes them interesting targets for drug development. Determination of the structure of these receptors will help to design more specific...

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Detalhes bibliográficos
Publicado no:Front Pharmacol
Main Authors: Heydenreich, Franziska M., Vuckovic, Ziva, Matkovic, Milos, Veprintsev, Dmitry B.
Formato: Artigo
Idioma:Inglês
Publicado em: Frontiers Media S.A. 2015
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC4403299/
https://ncbi.nlm.nih.gov/pubmed/25941489
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3389/fphar.2015.00082
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