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Kinetic characterization of human butyrylcholinesterase mutants for hydrolysis of cocaethylene

It is known that majority of cocaine users also consume alcohol. Alcohol can react with cocaine to produce a significantly more cytotoxic compound, cocaethylene. Hence, a truly valuable cocaine-metabolizing enzyme for cocaine abuse/overdose treatment should be efficient for not only cocaine itself,...

Täydet tiedot

Tallennettuna:
Bibliografiset tiedot
Julkaisussa:Biochem J
Päätekijät: Hou, Shurong, Zhan, Max, Zheng, Xirong, Zhan, Chang-Guo, Zheng, Fang
Aineistotyyppi: Artigo
Kieli:Inglês
Julkaistu: 2014
Aiheet:
Linkit:https://ncbi.nlm.nih.gov/pmc/articles/PMC4371731/
https://ncbi.nlm.nih.gov/pubmed/24870023
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1042/BJ20140360
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