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Evidence for an Elevated Aspartate pK(a) in the Active Site of Human Aromatase

Aromatase (CYP19A1), the enzyme that converts androgens to estrogens, is of significant mechanistic and therapeutic interest. Crystal structures and computational studies of this enzyme shed light on the critical role of Asp(309) in substrate binding and catalysis. These studies predicted an elevate...

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Библиографические подробности
Опубликовано в: :J Biol Chem
Главные авторы: Di Nardo, Giovanna, Breitner, Maximilian, Bandino, Andrea, Ghosh, Debashis, Jennings, Gareth K., Hackett, John C., Gilardi, Gianfranco
Формат: Artigo
Язык:Inglês
Опубликовано: American Society for Biochemistry and Molecular Biology 2015
Предметы:
Online-ссылка:https://ncbi.nlm.nih.gov/pmc/articles/PMC4294484/
https://ncbi.nlm.nih.gov/pubmed/25425647
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1074/jbc.M114.595108
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