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Site-Specific Coupling and Sterically Controlled Formation of Multimeric Antibody Fab Fragments with Unnatural Amino Acids

Immunoconjugates and multispecific antibodies are rapidly emerging as highly potent experimental therapeutics against cancer. We have developed a method to incorporate an unnatural amino acid, p-acetylphenylalanine (pAcPhe) into an antibody antigen binding fragment (Fab) targeting HER2 (human epider...

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Bibliografiske detaljer
Udgivet i:J Mol Biol
Main Authors: Hutchins, Benjamin M., Kazane, Stephanie A., Staflin, Karin, Forsyth, Jane S., Felding-Habermann, Brunhilde, Schultz, Peter G., Smider, Vaughn V.
Format: Artigo
Sprog:Inglês
Udgivet: 2011
Fag:
Online adgang:https://ncbi.nlm.nih.gov/pmc/articles/PMC4278757/
https://ncbi.nlm.nih.gov/pubmed/21237172
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.jmb.2011.01.011
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