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Haplotype Variations in Glutathione Transferase Zeta 1 Influence the Kinetics and Dynamics of Chronic Dichloroacetate in Children

Dichloroacetate (DCA) is biotransformed by glutathione transferase zeta 1 (GSTZ1), a bifunctional enzyme that, as maleylacetoacetate isomerase (MAAI), catalyzes the penultimate step in tyrosine catabolism. DCA inhibits GSTZ1/MAAI, leading to delayed plasma drug clearance and to accumulation of poten...

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Détails bibliographiques
Publié dans:J Clin Pharmacol
Auteurs principaux: AL, Shroads, BS, Coats, CW, McDonough, T, Langaee, PW, Stacpoole
Format: Artigo
Langue:Inglês
Publié: 2014
Sujets:
Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC4276489/
https://ncbi.nlm.nih.gov/pubmed/25079374
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/jcph.371
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