Načítá se...

Identification of an inhibitor-binding site to HIV-1 integrase with affinity acetylation and mass spectrometry

We report a methodology that combines affinity acetylation with MS analysis for accurate mapping of an inhibitor-binding site to a target protein. For this purpose, we used a known HIV-1 integrase inhibitor containing aryl di-O-acetyl groups (Acetylated-Inhibitor). In addition, we designed a control...

Celý popis

Uloženo v:
Podrobná bibliografie
Hlavní autoři: Shkriabai, Nick, Patil, Sachindra S., Hess, Sonja, Budihas, Scott R., Craigie, Robert, Burke, Terrence R., Le Grice, Stuart F. J., Kvaratskhelia, Mamuka
Médium: Artigo
Jazyk:Inglês
Vydáno: National Academy of Sciences 2004
Témata:
On-line přístup:https://ncbi.nlm.nih.gov/pmc/articles/PMC406438/
https://ncbi.nlm.nih.gov/pubmed/15118107
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1073/pnas.0400873101
Tagy: Přidat tag
Žádné tagy, Buďte první, kdo otaguje tento záznam!