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Hypoxia-selective O(6)-Alkylguanine-DNA Alkyltransferase Inhibitors: Design, Synthesis and Evaluation of 6-(Benzyloxy)-2-(aryldiazenyl)-9H-purines as Prodrugs of O(6)-Benzylguanine

O(6)-Alkylguanine-DNA alkyltransferase (AGT) is a DNA repair protein which removes alkyl groups from the O-6 position of guanine, thereby providing strong resistance to anticancer agents which alkylate this position. The clinical usefulness of these anticancer agents would be substantially augmented...

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Detalhes bibliográficos
Main Authors: Zhu, Rui, Baumann, Raymond P., Penketh, Philip G., Shyam, Krishnamurthy, Sartorelli, Alan C.
Formato: Artigo
Idioma:Inglês
Publicado em: 2013
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC3722860/
https://ncbi.nlm.nih.gov/pubmed/23311288
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jm301804p
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